TSIPROTERON (Cyproterone). 6-Chloro-1 b, 2-hydroxy-3 digidro-17- 'H cyclone promoted [1, 2] pregna-1, 4, 6 trien-3, 20-dionatsetat.

     Synonyms: Androkur, Androcur, Cyprostat, Cyproteronacetat.

     Tsiproteronatsetat is antiandrogenom steroidnoy structure. Oppressing education complex HSBG with androgenovymi kletkah- receptors in the target, including in the nuclei of cancer cells prostate gland. Oppressing also release gonadotropinov and thus delaying the effect of endogenous testosterone on the tumor cells.

     Apply tsiproteronatsetat with inoperable cancer of prostate gland. Sometimes effective in tumor resistance to other hormonal drugs.

     Sometimes tsiproteronatsetat apply to women with severe forms giperandrogennoy activity (girsutizm heavy, heavy androgenozavisimaya loss, severe acne and oily), as well as premature sexual development in children.

     Inside accepted as tablets after eating, vine liquid.

     Normal starting dose for men and 1 tablet (50 mg) two times a day. If necessary to increase the dose of 2 tablets 2 to 3 times a day. After therapeutic benefits to reduce the dose of 1 - 0.5 tablets per day.

     Women are usually appointed to 1 tablet (50 mg) two times a day.

     Children are at 0.5-2 1 tablet twice a day.

     Men in the application of the drug may develop ginekomastii, pain in the milk glands. Women may oppression ovulation.

     Using large doses may breach liver function, the delay fluid in the body.

     When pregnancy application tsiproteronatsetata counter.

     Please note that the typical low tsiproteronatsetatu androgennaya activity, which is wary of the risk of cancer in the prostate gland. Therefore, the recent preference for non-steroid antiandrogenam.

     Form release: pills to 0.05 g (50 mg) in a package of 50 pieces.

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